
Journal of Enzyme Inhibition and Medicinal Chemistry p. 397 - 400 (2014)
Update date:2022-07-29
Topics:
Shimada, Hideaki
Tanigawa, Takahiro
Matayoshi, Kazunori
Katakura, Kazufumi
Babazono, Ken
Takayama, Hiroyuki
Murahashi, Tsuyoshi
Akita, Hiroyuki
Higuchi, Toshiyuki
Eto, Masashi
Imamura, Yorishige
Context and objective: The present study is to elucidate the comparative inhibition of tetrameric carbonyl reductase (TCBR) activity by alkyl 4-pyridyl ketones, and to characterize its substrate-binding domain. Materials and methods: The inhibitory effect
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