Journal of Medicinal Chemistry p. 7741 - 7753 (2018)
Update date:2022-08-15
Topics:
Fu, Haigen
Zhang, Jielin
Tepper, Pieter G.
Bunch, Lennart
Jensen, Anders A.
Poelarends, Gerrit J.
Aspartate (Asp) derivatives are privileged compounds for investigating the roles governed by excitatory amino acid transporters (EAATs) in glutamatergic neurotransmission. Here, we report the synthesis of various Asp derivatives with (cyclo)alkyloxy and (
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