Bioorganic and Medicinal Chemistry Letters p. 1401 - 1405 (2005)
Update date:2022-08-02
Topics:
Duffy, Joseph L.
Kirk, Brian A.
Konteatis, Zenon
Campbell, Elizabeth L.
Liang, Rui
Brady, Edward J.
Candelore, Mari Rios
Ding, Victor D.H.
Jiang, Guoqiang
Liu, Frank
Qureshi, Sajjad A.
Saperstein, Richard
Szalkowski, Deborah
Tong, Sharon
Tota, Lauri M.
Xie, Dan
Yang, Xiaodong
Zafian, Peter
Zheng, Song
Chapman, Kevin T.
Zhang, Bei B.
Tata, James R.
A novel class of antagonists of the human glucagon receptor (hGCGR) has been discovered. Systematic modification of the lead compound identified substituents that were essential for activity and those that were amenable to further optimization. This SAR e
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