Potential synthetic codeine substitutes: (-)-3-O-aryl-N-methylmorphinans

DOI: 10.1021/jm00375a024

Source and publish data:

Journal of Medicinal Chemistry p. 1219 - 1222 (1984)

Update date:2022-07-30

Topics:

Authors:

Mohacsi Mohacsi

Hayes Hayes

Spinwall

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Article abstract of DOI:10.1021/jm00375a024

A series of novel O-aryl-N-methylmorphinans were synthesized by the Ullmann reaction from levorphanol in our search for a synthetic codeine substitute with reduced addition liability. The compounds were evaluated for antinociceptive potency and receptor b

Full text of DOI:10.1021/jm00375a024

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