Divergent Synthesis of 1H-Indazoles and 1H-Pyrazoles from Hydrazones via Iodine-Mediated Intramolecular Aryl and sp3 C–H Amination

DOI: 10.1002/adsc.201700824

Source and publish data:

Advanced Synthesis and Catalysis p. 3378 - 3387 (2017)

Update date:2022-07-30

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Authors:

Wei, Wei

Wang, Zhen

Yang, Xikang

Yu, Wenquan

Chang, Junbiao

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Article abstract of DOI:10.1002/adsc.201700824

A divergent intramolecular C–H amination of hydrazones has been developed employing molecular iodine (I₂) as the sole oxidant. The required hydrazone substrates were readily obtained by condensation of hydrazines with the corresponding ketones.

Full text of DOI:10.1002/adsc.201700824

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