
Biochemical Pharmacology p. 63 - 72 (2016)
Update date:2022-08-05
Topics:
Read, Cai
Fitzpatrick, Christopher M.
Yang, Peiran
Kuc, Rhoda E.
Maguire, Janet J.
Glen, Robert C.
Foster, Richard E.
Davenport, Anthony P.
Apelin peptide analogues displaying bias towards G protein signalling pathways have beneficial cardiovascular actions compared with the native peptide in humans in vivo. Our aim was to determine whether small molecule agonists could retain G protein bias.
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