Bioorganic and Medicinal Chemistry Letters p. 5709 - 5712 (2004)
Update date:2022-08-05
Topics:
Romagnoli, Romeo
Baraldi, Pier Giovanni
Pavani, Maria Giovanna
Tabrizi, Mojgan Aghazadeh
Moorman, Allan R.
Di Virgilio, Francesco
Cattabriga, Elena
Pancaldi, Cecilia
Gessi, Stefania
Borea, Pier Andrea
The design, synthesis, and preliminary biological evaluation of the first potent radioligand antagonist for the P2X7 receptor, named [ 3H]-1-[(S)-N,O-bis-(isoquinolinesulfonyl)-N-methyl-tyrosyl] -4-(o-tolyl)-piperazine (compound 13),
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(2004)