4,5,6,7-Tetrahydroisothiazolo[5,4-c]pyridin-3-ol and related analogues of THIP. Synthesis and biological activity

DOI: 10.1021/jm00360a020

Source and publish data:

Journal of Medicinal Chemistry p. 895 - 900 (1983)

Update date:2022-08-02

Topics:

Authors:

Krogsgaard-Larsen

Mikkelsen

Jacobsen

Falch Falch

Curtis Curtis

Peet Peet

Leah Leah

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Article abstract of DOI:10.1021/jm00360a020

The thio analogues of the GABA (γ-aminobutyric acid) agonist THIP (4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-3-ol), the GABA uptake inhibitor THPO (4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-3-ol), and the glycine antagonist THAZ (5,6,7,8-tetrahydro-4H-is

Full text of DOI:10.1021/jm00360a020

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