Bioorganic and Medicinal Chemistry Letters p. 3149 - 3152 (2002)
Update date:2022-08-03
Topics:
Wang, Yuguang
Chackalamannil, Samuel
Hu, Zhiyong
Boyle, Craig D.
Lankin, Claire M.
Xia, Yan
Xu, Ruo
Asberom, Theodros
Pissarnitski, Dmitri
Stamford, Andrew W.
Greenlee, William J.
Skell, Jeffrey
Kurowski, Stanley
Vemulapalli, Subbarao
Palamanda, Jairam
Chintala, Madhu
Wu, Ping
Myers, Joyce
Wang, Peng
We have discovered potent and selective xanthine PDE5 inhibitors. Compound 25 (PDE5 IC50=0.6 nM, PDE6/PDE5=101) demonstrated similar functional efficacy and PK profile to Sildenafil (PDE5 IC50=3.5 nM, PDE6/PDE5=7).
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Doi:10.1039/a706802f
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