Bioorganic and Medicinal Chemistry Letters p. 2051 - 2056 (2016)
Update date:2022-08-03
Topics:
Lan, Yu
Songyang, Yiyan
Zhang, Lingli
Peng, Yan
Song, Jinchun
The synthesis and biological evaluation of new series of 6,7-dihydro-5H-cyclopenta[d]pyrimidine and 5,6,7,8-tetrahydroquinazoline derivatives as selective sigma-1 receptor (σ1R) antagonists are reported. The receptor affinities of new compounds
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