European Journal of Medicinal Chemistry (2020)
Update date:2022-08-02
Topics:
Xiao, Ting
Tang, Jia-Fan
Meng, Ge
Pannecouque, Christophe
Zhu, Yuan-Yuan
Liu, Gen-Yan
Xu, Zhi-Qiang
Wu, Feng-Shou
Gu, Shuang-Xi
Chen, Fen-Er
A series of indazolyl-substituted piperidin-4-yl-aminopyrimidines (IPAPYs) were designed from two potent HIV-1 NNRTIs piperidin-4-yl-aminopyrimidine 3c and diaryl ether 4 as the lead compounds by molecular hybridization strategy. The target molecules 5a-q
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