A Synthesis of Optically Active 4-Diethoxyphosphinyl-3-(1-hydroxyethyl)-2-azetidinone: A Potential Precursor to (1-Aminoalkyl)-phosphonic Acid Derivatives

DOI: 10.1246/bcsj.60.645

Source and publish data:

Bulletin of the Chemical Society of Japan p. 645 - 648 (1987)

Update date:2022-07-29

Topics:

Authors:

Shiozaki, Masao

Masuko, Hidekazu

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1246/bcsj.60.645

Optically active 4-diethoxyphosphinyl-3-(1-hydroxyethyl)-2-azetidinone (8) was synthesized from (2R,3R)-N-diethoxyphosphinylmethyl-2,3-epoxybutyramide derivatives, and compound 8 was alternatively synthesized from (3R,4R)-4-acetoxy-3-<(R)-1-(t-butyldimeth

Full text of DOI:10.1246/bcsj.60.645

Products guided by the article

Product name:(2S,3R)-N-(diethoxyphosphinylmethyl)-N-(4-methoxybenzyl)-2-bromo-3-hydroxybutyramide

Cas No:93591-34-5

R&D Labs maybe for 93591-34-5

Hangzhou JINLAN Pharm-Drugs Technology Co., Ltd

website:http://www.jlpharms.com

Contact:+86-571-86982636

Address:Rm A606, Fuyi Center, jianqiao street, Jianggan Area
Xi'an Tizan Tech & Industry Co., Ltd.

Contact:86-18629066522

Address:C3009 TANG FENG INTERNATIONAL PLAZA, NO.18 FENGHUI NAN ROAD, XI'AN HIGH TECH ZONE, 710075 CHINA.
Jiangxi Dongbang Pharmaceutical Co., Ltd.

Contact:+86-795-4433603, 4433388

Address:Fengxin Industrial Park, Fengxin County, Jiangxi Province, P.R.C
Wuhan Shengmao Corp

website:http://www.shengmaochem.com

Contact:86-27-82853423, 82819281

Address:Rm 202, A Unit Huaqiao Building No. 2, Lihuangpi Road, Wuhan, China
Lanzhou huibang biological chemical technology Co., LTD

Contact:0931-7843964

Address:NO.2011,Yannan Road,Chengguan,

Relevant to this article

The chemistry of drugs. Part IV. Configurations of antimalarials derived from qinghaosu: dihydroqinghaosu, artemether, and artesunic acid

Doi:10.1002/hlca.19840670615
(1984)
DEUTERIUM ISOTOPE EFFECTS IN THE META PHOTOCYCLOADDITION OF AROMATIC COMPOUNDS TO ALKENES

Doi:10.1016/S0040-4039(00)98745-8
(1985)
Kinetic and labeling studies of the formation and trapping reactions of dimethylgermylene

Doi:10.1021/om00110a004
(1989)
Synthesis and biological evaluation of novel glycosyl-containing 1,2,4-triazolo[3,4-b][1,3,4]thiadiazole derivatives as acetylcholinesterase inhibitors

Doi:10.3184/174751917X15064232103047
(2017)
Antinociceptive effect of 3-(2,3-dimethoxyphenyl)-1-(5-methylfuran-2-yl)prop-2-en-1-one in mice models of induced nociception

Doi:10.3390/molecules21081077
(2016)
DICHLORO-BIS(TRIFLUOROMETHANESULFONATO)TITANIUM(IV) AS AN EFFECTIVE PROMOTER IN THE CLAISEN ESTER CONDENSATION

Doi:10.1246/cl.1984.1867
(1984)

Article Doi