Studies on analgesic oligopeptides. III. Synthesis and analgesic activity after subcutaneous administration of [D-Arg2]dermorphin and its N-terminal tetrapeptide analogs

DOI: 10.1248/cpb.33.1528

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1528 - 1536 (1985)

Update date:2022-08-02

Topics:

Authors:

Sasaki Sasaki

Matsui Matsui

Fujita Fujita

Hosono Hosono

Taguchi Taguchi

Suzuki Suzuki

Sakurada

Sato Sato

Sakurada

Kisara Kisara

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.33.1528

[D-Arg²]dermorphin and nineteen N-terminal tetrapeptide analogs were synthesized by a conventional solution method and their analgesic activities after subcutaneous administration to mice were examined. The analgesic effect was assessed by mean

Full text of DOI:10.1248/cpb.33.1528

NII-Electronic Library Service

Products guided by the article

Product name:H-Tyr-D-Arg-Phe(NO₂)-Gly-OEt

Cas No:99592-87-7

R&D Labs maybe for 99592-87-7

Dragon Chemical Co., Ltd.

Contact:0571-

Address:zhejing
Jinan Finer Chemical Co., Ltd

website:http://www.finerchem.com

Contact:+86-531-88989536

Address:New Material Industry Park, Jinan Ciyt, China
Beijing Chemdow Co., Ltd

website:http://www.chemdow.com

Contact:0086-10-82435335

Address:Room 401,Unit 3,4th Floor,Shangdijiayuan,Shangdi East Road, Haidian District,Beijing
LIANYUNGANG YC FINE CHEMICAL CO., LTD

Contact:+86-518-858 99188

Address:Shangdong Modern Bldg, South Greenpark Road, Lianyungang, Jiangsu Pro. China
Zhuhai Rundu Pharmaceutical co.,Ltd

Contact:+86-756-7630755

Address:No.6,North Airport Road,Sanzao Town,Jinwan District

Relevant to this article

A Novel Cycloaddition Reaction for Obtaining 1H-Indoles from 3-(α,β-Unsaturated alkenyl)phenols

Doi:10.1021/jo00066a031
(1993)
SELENYL CHLORIDE AS AN ACTIVE CHLORINATING AGENT

Doi:10.1007/BF00953371
(1986)
Hydration of Diacetylene Compounds. Synthesis of a Marine Natural Product: (+/-)-1-(2,6,6-Trimethyl-4-hydroxycyclohexenyl)-1,3-butanedione

Doi:10.1021/jo00353a022
(1986)
Doi:10.1002/ardp.19582910210
(1958)
Microwave-assisted silica-supported aluminum chloride-catalyzed Friedel-Crafts alkylation

Doi:10.1016/j.tetlet.2012.07.131
(2012)
Sterically congested macrobicycles with heteroatomic bridgehead functionality

Doi:10.1016/j.tet.2013.10.018
(2013)

Article Doi