Studies on analgesic oligopeptides. III. Synthesis and analgesic activity after subcutaneous administration of [D-Arg2]dermorphin and its N-terminal tetrapeptide analogs

DOI: 10.1248/cpb.33.1528

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1528 - 1536 (1985)

Update date:2022-08-02

Topics:

Authors:

Sasaki Sasaki

Matsui Matsui

Fujita Fujita

Hosono Hosono

Taguchi Taguchi

Suzuki Suzuki

Sakurada

Sato Sato

Sakurada

Kisara Kisara

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.33.1528

[D-Arg²]dermorphin and nineteen N-terminal tetrapeptide analogs were synthesized by a conventional solution method and their analgesic activities after subcutaneous administration to mice were examined. The analgesic effect was assessed by mean

Full text of DOI:10.1248/cpb.33.1528

NII-Electronic Library Service

Products guided by the article

Product name:H-Tyr-D-Arg-Phe(NO₂)-Gly-OEt

Cas No:99592-87-7

R&D Labs maybe for 99592-87-7

Jiangsu Feymer Technology Co., Ltd.

Contact:+86-512-58110132

Address:Fenghuang Town, Zhangjiagang City, Jiangsu Province, China
Kaiping Genuine Biochemical Pharmaceutical Co.,Ltd.

Contact:+86-750-2881198

Address:No.1, Xinke Road, Shatang Town, Kaiping, Guangdong Province, P.R.China
A-Chem Technologies Co.,Ltd.

Contact:+86-512-69561895

Address:No.111, Building A4, 218 Xinghu Street, Suzhou Industrial Park, P. R. China
Chengdu Green Young Biopharmaceutical INC

Contact:+86-28-85337952

Address:1-B-26,Tianhe Industry Park, No.1480 of Tianfu Road,Chengdu,P.R.China,610000
JIEJIE GROUP CO.,LTD.

Contact:+86 021-51698675

Address:1701, Jielong Plaza, No.618 Pingliang Rd, ShangHai,China

Relevant to this article

A Novel Cycloaddition Reaction for Obtaining 1H-Indoles from 3-(α,β-Unsaturated alkenyl)phenols

Doi:10.1021/jo00066a031
(1993)
SELENYL CHLORIDE AS AN ACTIVE CHLORINATING AGENT

Doi:10.1007/BF00953371
(1986)
Hydration of Diacetylene Compounds. Synthesis of a Marine Natural Product: (+/-)-1-(2,6,6-Trimethyl-4-hydroxycyclohexenyl)-1,3-butanedione

Doi:10.1021/jo00353a022
(1986)
Doi:10.1002/ardp.19582910210
(1958)
Microwave-assisted silica-supported aluminum chloride-catalyzed Friedel-Crafts alkylation

Doi:10.1016/j.tetlet.2012.07.131
(2012)
Sterically congested macrobicycles with heteroatomic bridgehead functionality

Doi:10.1016/j.tet.2013.10.018
(2013)

Article Doi