Studies on analgesic oligopeptides. III. Synthesis and analgesic activity after subcutaneous administration of [D-Arg2]dermorphin and its N-terminal tetrapeptide analogs

DOI: 10.1248/cpb.33.1528

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1528 - 1536 (1985)

Update date:2022-08-02

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Authors:

Sasaki Sasaki

Matsui Matsui

Fujita Fujita

Hosono Hosono

Taguchi Taguchi

Suzuki Suzuki

Sakurada

Sato Sato

Sakurada

Kisara Kisara

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Article abstract of DOI:10.1248/cpb.33.1528

[D-Arg²]dermorphin and nineteen N-terminal tetrapeptide analogs were synthesized by a conventional solution method and their analgesic activities after subcutaneous administration to mice were examined. The analgesic effect was assessed by mean

Full text of DOI:10.1248/cpb.33.1528

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