
Bioorganic and Medicinal Chemistry Letters p. 2906 - 2909 (2005)
Update date:2022-08-17
Topics:
Fonvielle
Mariano
Therisod
We describe the synthesis and evaluation of three new competitive inhibitors of triose-phosphate isomerase. One of them (phosphoglycoloamidoxime: Ki = 4.5 μM) is among the best reversible inhibitors so far reported for this enzyme.
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