Journal of Medicinal Chemistry p. 1247 - 1261 (2017)
Update date:2022-08-17
Topics:
Harris, Philip A.
Berger, Scott B.
Jeong, Jae U.
Nagilla, Rakesh
Bandyopadhyay, Deepak
Campobasso, Nino
Capriotti, Carol A.
Cox, Julie A.
Dare, Lauren
Dong, Xiaoyang
Eidam, Patrick M.
Finger, Joshua N.
Hoffman, Sandra J.
Kang, James
Kasparcova, Viera
King, Bryan W.
Lehr, Ruth
Lan, Yunfeng
Leister, Lara K.
Lich, John D.
MacDonald, Thomas T.
Miller, Nathan A.
Ouellette, Michael T.
Pao, Christina S.
Rahman, Attiq
Reilly, Michael A.
Rendina, Alan R.
Rivera, Elizabeth J.
Schaeffer, Michelle C.
Sehon, Clark A.
Singhaus, Robert R.
Sun, Helen H.
Swift, Barbara A.
Totoritis, Rachel D.
Vossenk?mper, Anna
Ward, Paris
Wisnoski, David D.
Zhang, Daohua
Marquis, Robert W.
Gough, Peter J.
Bertin, John
RIP1 regulates necroptosis and inflammation and may play an important role in contributing to a variety of human pathologies, including immune-mediated inflammatory diseases. Small-molecule inhibitors of RIP1 kinase that are suitable for advancement into
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