A route to dipeptides containing β-amino-α-hydroxy acid fragments by coupling of N-boc-β-lactams with α-amino esters. Application to the synthesis of (-)-bestatin

DOI: 10.1039/c39940001957

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 1957 - 1958 (1994)

Update date:2022-08-11

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Authors:

Palomo Palomo

Aizpurua

Cuevas Cuevas

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Article abstract of DOI:10.1039/c39940001957

α-Amino esters are smoothly acylated by N-Boc-3-alkoxy-4-alkyl-β-lactams in DMF under the influence of sodium azide, giving a novel dipeptide coupling reaction.

Full text of DOI:10.1039/c39940001957

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