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References
Antimicrobial resistance: report on global surveillance.; World Health Organization:
France, 2014.
2. Antimicrobial Resistance: Tackling a crisis for the health and wealth of nations.; The
Review on Antimicrobial Resistance: London, 2014.
1.
3
1
4
.
Tenover, F. C., Mechanisms of Antimicrobial Resistance in Bacteria. Am. J. Med. 2006,
19, (6, Supplement 1), S3-S10.
Blair, J. M. A.; Webber, M. A.; Alison J. Baylay; Ogbolu, D. O.; Piddock, L. J. V.,
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
.
Molecular mechanisms of antibiotic resistance. Nat. Rev. Microbiol. 2015, 13, 42-51.
5. Brogden, Antimicrobial peptides: pore formers or metabolic inhibitors in bacteria? Nat.
Rev. Microbiol. 2005, 3, 238-250.
6
3
7
.
Zasloff, M., Antimicrobial peptides of multicellular organisms. Nature 2002, 415, (6870),
89-95.
.
Jenssen, H. v.; Hamill, P.; Hancock, R. E. W., Peptide Antimicrobial Agents. Clin.
Microbiol. Rev. 2006, 19, (3), 491-511.
Hancock, R. E.; Sahl, H. G., Antimicrobial and host-defense peptides as new anti-
infective therapeutic strategies. Nat. Biotechnol. 2006, 24, (12), 1551-7.
Culf, A. S.; Ouellette, R. J., Solid-phase synthesis of N-substituted glycine oligomers
alpha-peptoids) and derivatives. Molecules 2010, 15, (8), 5282-335.
10. Giuliani, A.; Rinaldi, A. C., Beyond natural antimicrobial peptides: multimeric peptides
and other peptidomimetic approaches. Cell Mol. Life Sci. 2011, 68, (13), 2255-66.
1. Zuckermann, R. N.; Kerr, J. M.; Kent, S. B. H.; Moos, W. H., Efficient method for the
8.
9.
(
1
preparation of peptoids [oligo(N-substituted glycines)] by submonomer solid-phase synthesis. J.
Am. Chem. Soc. 1992, 114, (26), 10646-10647.
12.
Chongsiriwatana, N. P.; Wetzler, M.; Barron, A. E., Functional synergy between
antimicrobial peptoids and peptides against Gram-negative bacteria. Antimicrob. Agents
Chemother. 2011, 55, (11), 5399-402.
13.
Kapoor, R.; Eimerman, P. R.; Hardy, J. W.; Cirillo, J. D.; Contag, C. H.; Barron, A. E.,
Efficacy of antimicrobial peptoids against Mycobacterium tuberculosis. Antimicrob. Agents
Chemother. 2011, 55, (6), 3058-62.
14. Kapoor, R.; Wadman, M. W.; Dohm, M. T.; Czyzewski, A. M.; Spormann, A. M.;
Barron, A. E., Antimicrobial peptoids are effective against Pseudomonas aeruginosa biofilms.
Antimicrob Agents Chemother. 2011, 55, (6), 3054-7.
Chongsiriwatana, N. P.; Patch, J. A.; Czyzewski, A. M.; Dohm, M. T.; Ivankin, A.;
15.
Gidalevitz, D.; Zuckermann, R. N.; Barron, A. E., Peptoids that mimic the structure, function,
and mechanism of helical antimicrobial peptides. Proc. Natl. Acad. Sci. U S A 2008, 105, (8),
2794-9.
1
6.
Soc. 2003, 125, (40), 12092-3.
7. Hein-Kristensen, L.; Knapp, K. M.; Franzyk, H.; Gram, L., Bacterial membrane activity
Patch, J. A.; Barron, A. E., Helical peptoid mimics of magainin-2 amide. J. Am. Chem.
1
of alpha-peptide/beta-peptoid chimeras: influence of amino acid composition and chain length on
the activity against different bacterial strains. BMC Microbiol. 2011, 11, 144.
18.
Kennedy, J. P.; Williams, L.; Bridges, T. M.; Daniels, R. N.; Weaver, D.; Lindsley, C.
W., Application of Combinatorial Chemistry Science on Modern Drug Discovery. J. Comb.
Chem. 2008, 10, (3), 345-354.
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