International Journal of Pharmaceutics p. 48 - 57 (2019)
Update date:2022-08-29
Topics:
Sun, Jing
Yang, Dan
Cui, Shi-He
Zhang, Hai-Tao
Fu, Yu
Wang, Jian-Cheng
Zhang, Qiang
Gemcitabine (Gem) as an anti-cancer agent has been limited by its short circulation time and rapid metabolism that reflects in low tumor uptake and low therapeutic efficiency. To improve its anti-tumor activity, a novel FAPα enzyme-activated prodrug of Z-
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