SYNTHETIC STUDIES IN THE QUASSINOID SERIES. CONVERSION OF CHAPARRIN INTO CASTELANONE AND QUASSINOID ANALOGS.

DOI: 10.1016/S0040-4039(00)87397-9

Source and publish data:

Tetrahedron Letters p. 2567 - 2570 (1982)

Update date:2022-08-29

Topics:

Authors:

Caruso, Andrew J.

Polonsky, Judith

Rodriguez, Bertha Soto

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Article abstract of DOI:10.1016/S0040-4039(00)87397-9

Inactive chaparrin 1 has been converted in seven steps and 16 percent overall yield to castelanone 3 which is known to inhibit significantly growth of the murine lymphocytic leukemia P-388 cell line.The methodology developed has been applied to the preparation of quassinoid analogs 15, 16 and 17.

Full text of DOI:10.1016/S0040-4039(00)87397-9

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