(S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate

Base Information

• Chemical Name: (S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate
• CAS No.: 1004524-42-8
• Molecular Formula: C₁₇H₂₆BNO₅
• Molecular Weight: 335.208

Synonyms:(S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate

Chemical Property of (S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate

Chemical Property:

Purity/Quality:

99% ^*data from raw suppliers

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Technology Process of (S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate

There total 6 articles about (S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

(S)-methyl 2-((tert-butoxycarbonyl)amino)-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate (675832-36-7) → (S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate (1004524-42-8)

Guidance literature:

With trifluoroacetic acid; In dichloromethane; at 20 ℃;

Reference yield:

(S)-N-benzyloxycarbonyl-3-(4-methoxy-3-(4,4,5,5-tetramethyl[1,3,2]dioxaborolan-2-yl)phenyl)alanine methyl ester (353520-75-9) → (S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate (1004524-42-8)

Guidance literature:

With hydrogen; palladium on activated charcoal; In ethanol; under 760.051 Torr;

DOI:10.1021/ja073340u

Reference yield:

hydrogen (1333-74-0) + (S)-N-benzyloxycarbonyl-3-(4-methoxy-3-(4,4,5,5-tetramethyl[1,3,2]dioxaborolan-2-yl)phenyl)alanine methyl ester (353520-75-9) → (S)-methyl 2-amino-3-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)phenyl)propanoate (1004524-42-8)

Guidance literature:

With palladium on activated charcoal; In ethanol; treatment of boron compd. with H2 in 95% ethanol in presence of palladium catalyst;

DOI:10.1021/ja073340u

upstream raw materials:

(S)-N-benzyloxycarbonyl-3-(4-methoxy-3-(4,4,5,5-tetramethyl[1,3,2]dioxaborolan-2-yl)phenyl)alanine methyl ester

hydrogen

(S)-N-(tert-butoxycarbonyl)tyrosine methyl ester

(S)-methyl 2-((tert-butoxycarbonyl)amino)-3-(4-methoxyphenyl)propanoate

Downstream raw materials:

MeOC₆H₃ICH(NHBoc)CONHCH(CH₃)CONHCH(COOMe)CH₂C₆H₃(B(pinacolato))OMe

C₄₃H₅₅N₅O₁₁

(6S,9S,12S)-methyl 6-(3-iodo-4-methoxyphenyl)-1 2-(4-methoxy-3-(4,4,5 ,5-tetramethyl-1,3 ,2-dioxaborolan-2-yl)benzyl)-2,2,5 ,9-tetramethyl-4,7, 1 0-trioxo-3-oxa-5 ,8,11-triazatridecan-13-oate

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