111462-38-5Relevant articles and documents
Total synthesis and the anticancer activity of (+)-spisulosine
Fabi?íková, Milica,Martinková, Miroslava,Hirková, Simona,Gonda, Jozef,Pilátová, Martina Bago,G?nciová, Gabriela
, p. 26 - 36 (2016/10/04)
The total synthesis of the anticancer agent (+)-spisulosine has been accomplished. The strategy involved a substrate-controlled aza-Claisen rearrangement to establish the erythro-configured amino-alcohol motif followed by deoxygenation to create a methyl
CYCLIC SULFONIUM SALT, PROCESS FOR PRODUCTION OF SAME, AND alpha-GLUCOSIDASE INHIBITOR COMPRISING SAME
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Paragraph 0090-0092, (2014/01/08)
Provided is a novel cyclic sulfonium salt compound which is useful for the prevention or treatment of diabetes and the like. The present invention relates to a novel cyclic sulfonium salt compound represented by general formula (I) or (II), an isomer or solvate of the compound, or a pharmaceutically acceptable salt of the compound or the isomer or solvate. The present invention also relates to an α-glucosidase inhibitor, a pharmaceutical composition for preventing or treating diabetes, and an anti-diabetes food, each of which comprises the compound represented by general formula (I) or (II) and the like.
The formal synthesis of 3-epi jaspine B using stereoselective intramolecular oxa-Michael addition
Rao, G. Srinivas,Sudhakar, Neela,Rao, B. Venkateswara,Basha, S. Jeelani
experimental part, p. 1963 - 1970 (2010/10/18)
The formal synthesis of 3-epi jaspine B was achieved by using a stereoselective intramolecular oxa-Michael addition. The diacetate derivative of 3-epi jaspine B was also synthesized.