1145-57-9Relevant academic research and scientific papers
SUBSTITUTED 4-ARYLOXY AND 4-ARYLSULFANYL-PHENYL-2-AMINOTHIAZOLES AS INHIBITORS OF CELL PROLIFERATION
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Page/Page column 30-33, (2008/06/13)
The invention discloses compounds which are substituted 4-aryloxy and 4-arylsulfanyl-phenyl-2-aminothiazoles with anti-cancer activity. The invention futher discloses methods of preparing compounds of the invention. The invention also discloses methods of inhibiting cell proliferation and tumor growth in a subject by administering compounds of the invention to the subject.
Synthesis and evaluation of substituted 4-aryloxy- and 4-arylsulfanyl- phenyl-2-aminothiazoles as inhibitors of human breast cancer cell proliferation
Gorczynski, Michael J.,Leal, Rachel M.,Mooberry, Susan L.,Bushweller, John H.,Brown, Milton L.
, p. 1029 - 1036 (2007/10/03)
Several substituted 4-aryloxy- and 4-arylsulfanyl-phenyl-2-aminothiazoles were synthesized and evaluated for cytotoxic activity against estrogen-positive, estrogen-negative, and adriamycin-resistant human breast cancer cell lines. 4-[4′-(3,4-Dichlorophenoxy)-phenyl]-thiazol-2-yl ammonium iodide demonstrated potent activity against both estrogen-positive and negative breast cancer cell lines with low micromolar (μM) GI50 values. In addition, we have identified several 2-aminothiazoles that demonstrated selective potency for the adriamycin-resistant and estrogen-negative breast cancer cell lines. The results suggest that these 2-aminothiazoles represent lead compounds for evaluation in animal models of breast cancer.
SYNTHESIS AND REACTIVITY OF ARYLOXYCUMENYL CHLORIDES
Litvinenko, L. M.,Benndorf, V.,Popova, R. S.,Popov, A. F.,Tormosin, I. I.
, p. 680 - 683 (2007/10/02)
A series of derivatives of aryloxycumenyl chlorides containing substituents (methyl, methoxy, fluorine, and chlorine) at positions 3 and 4 of the aryl ring were synthesized.From the results from their solvolysis in 90 vol. percent aqueous acetone it was concluded that there is strong transfer of the electronic effects through the diphenyl ether system comparable with that in biphenyl.
