139975-99-8

Upstream product

• 24424-99-5 di-tert-butyl dicarbonate 
• 132-86-5 1,3-dihydroxynaphthalene 
• 139975-98-7 tert-butyl-(4-hydroxynaphthalen-2-yl)carbamate 
• 129918-05-4 2--4-(benzyloxy)-1-bromonaphthalene 
• 122745-37-3 2-((tert-Butyloxycarbonyl)amino)-4-(benzyloxy)-1-bromonaphthalene 
• 122745-36-2 N-(tert-butyloxycarbonyl)-4-(benzyloxy)-2-naphthylamine 
• 56061-88-2 Triphenyl<(2-tetrahydropyranyloxy)methyl>phosphonium chloride 
• 129918-06-5 2--4-(benzyloxy)-1-bromonaphthalene 

Downstream Products

• 122745-39-5 5-(benzyloxy)-3-(tert-butyloxycarbonyl)-1-(hydroxymethyl)-1,2-dihydro-3H-benzindole 
• 139976-01-5 5-(Benzyloxy)-3-(tert-butyloxycarbonyl)-1-<(tetrahydropyranyloxy)methyl>-1,2-dihydro-3H-benzindole 

Relevant academic research and scientific papers

An Improved Synthesis of 1,2,9,9a-Tetrahydrocyclopropabenzindol-4-one (CBI): A Simplified Analogue of the CC-1065 Alkylation Subunit

A concise and improved synthesis of 11, the immediate precursor to N-BOC-CBI and related analogues of CC-1065 incorporating the 1,2,9,9a-tetrahydrocyclopropabenzindol-4-one alkylation subunit, is detailed based on a direct 5-exo-trig aryl radical-al