158250-56-7Relevant academic research and scientific papers
Chemoenzymatic syntheses of carbasugar analogues of nucleoside diphosphate sugars: UDP-carba-Gal, UDP-carba-GlcNAc, UDP-carba-Glc, and GDP-carba-Man
Seo, Kyung-Chang,Kwon, Young-Geol,Kim, Dae-Hee,Jang, In-Sook,Cho, Jin-Won,Chung, Sung-Kee
supporting information; experimental part, p. 1733 - 1735 (2009/08/08)
Chemoenzymatic syntheses of several NDP-carba-sugars have been successfully carried out, and these essential cofactor analogues are expected to be selective inhibitors of glycosyltransferase enzymes. The Royal Society of Chemistry.
The synthesis of a new class of potential inhibitors for glycoside hydrolases
Stick, Robert V.,Stubbs, Keith A.
, p. 529 - 547 (2007/10/03)
Some attempts toward the synthesis of novel inhibitors of glycosyl transferases are described. More successfully, the synthesis of an activated cyclopropacyclohexene and an amide and an amine of a cyclopropa-fused pyranose are described. None of these three novel compounds proved to be a significant inhibitor of a retaining α-glucosidase from barley. Copyright Taylor & Francis, Inc.
Carbohydrates to carbocycles: An expedient synthesis of pseudo-sugars
Sudha,Nagarajan
, p. 925 - 926 (2007/10/03)
A short and versatile synthesis of pseudo-sugars from sugars utilizing the Claisen rearrangement as the key step is described.
Synthesis and Glycosidase-inhibitory Activity of Cyclophellitol Analogues
Tai, Vincent W.-F.,Fung, P.-H.,Wong, Y.-S.,Shing, Tony K. M.
, p. 1353 - 1362 (2007/10/02)
The 6-deoxy-1,2-anhydro-analogues of cyclophellitol, 5 and 6, have been synthesised from diol 11 via regioselective ring opening of the cyclic sulfate 15, an internal SN2 reaction and hydrogenolysis.Compounds 5,6, cyclophellitol 1 and its diast
