192384-87-5Relevant articles and documents
Synthesis and in vitro binding studies of piperazine-alkyl-naphthamides: Impact of homology and sulphonamide/carboxamide bioisosteric replacement on the affinity for 5-HT1A, α2A, D4.2, D3 and D2L receptors
Résimont, Mélissa,Liégeois, Jean-Fran?ois
scheme or table, p. 5199 - 5202 (2010/10/03)
A series of carboxamide and sulphonamide alkyl(ethyl to hexyl)piperazine analogues were prepared and tested for their affinity to bind to a range of receptors potentially involved in psychiatric disorders. These chemical modifications led us to explore th
2-NAPHTHAMIDE DERIVATIVES AND THEIR THERAPEUTIC APPLICATIONS
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, (2008/06/13)
The invention related to 2-naphthamide derivatives, in the form of bases or of salts, corresponding to the following general formula (I): STR1 in which: the Z--Y entity represents an N--CH 2, C= CH or CH--CH. sub.2 group;R 1 represents a hydrogen, f