55468-69-4Relevant academic research and scientific papers
9-AMINOACRIDINE DERIVATIVES, THEIR PREPARATION AND USES
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Page/Page column 26-27, (2011/05/11)
N-substituted 9-aminoacridine and bis-acridino derivatives containing electron- withdrawing groups (EWG) or electron-donating groups (EDG), including amino acid residues, and one-pot methods for their synthesis are disclosed. The derivatives are potential
One-pot derivatization of medicinally important 9-aminoacridines by reductive amination and SNAr reaction
Gellerman, Gary,Gaisin, Vladimir,Brider, Tamara
experimental part, p. 836 - 839 (2010/03/04)
A new highly efficient one-pot derivatization of medicinally important 9-aminoacridines (9-AA) at the amine position is described. Simple reductive amination and SNAr reaction using easily accessible starting materials give a fast entry to novel 9-AA derivatives for biological screening.
