Amino acids and peptides. XXIII. Leu-enkephalin analoges containing a fluorinated amino acid at position 2, 4 or 5

DOI: 10.1248/cpb.42.1658

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1658 - 1662 (1994)

Update date:2022-09-26

Topics:

Authors:

Maeda Maeda

Kawasaki

Taguchi Taguchi

Kobayashi

Yamamoto

Shimokawa

Takahashi

Nakao Nakao

Kaneto Kaneto

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Article abstract of DOI:10.1248/cpb.42.1658

Fluorinated analogs of Leu-enkephalin were synthesized by the solution method and the solid-phase method. The synthetic peptides were examined for opioid activities on mouse vas deferens and guinea pig ileum. Among the synthetic peptides, [D-Ala^{2
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Full text of DOI:10.1248/cpb.42.1658

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