A GENERAL PREPARATION OF FLUOROALLYLAMINE ENZYME INHIBITORS INCORPORATING A Β-SUBSTITUTED HETEROATOM

DOI: 10.1016/S0040-4039(00)89256-4

Source and publish data:

Tetrahedron Letters p. 3807 - 3810 (1985)

Update date:2022-07-30

Topics:

Authors:

McDonald, Ian A.

Bey, Philippe

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Article abstract of DOI:10.1016/S0040-4039(00)89256-4

A general route to β-heteroatom substituted fluoroallylamines is described.This has led to the synthesis of new time-dependent inhibitors of monoamine oxidase, diamine oxidase and γ-aminobutyric acid transaminase.

Full text of DOI:10.1016/S0040-4039(00)89256-4

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