A GENERAL PREPARATION OF FLUOROALLYLAMINE ENZYME INHIBITORS INCORPORATING A Β-SUBSTITUTED HETEROATOM

DOI: 10.1016/S0040-4039(00)89256-4

Source and publish data:

Tetrahedron Letters p. 3807 - 3810 (1985)

Update date:2022-07-30

Topics:

Authors:

McDonald, Ian A.

Bey, Philippe

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)89256-4

A general route to β-heteroatom substituted fluoroallylamines is described.This has led to the synthesis of new time-dependent inhibitors of monoamine oxidase, diamine oxidase and γ-aminobutyric acid transaminase.

Full text of DOI:10.1016/S0040-4039(00)89256-4

Products guided by the article

Product name:(Z)-3-Fluoro-2-phenylsulfanylmethyl-allylamine

Cas No:103362-76-1

R&D Labs maybe for 103362-76-1

Laohekou Jinghong Chemical Co.,Ltd

Contact:+86-0710-3702747

Address:163.East，Huagong Road，Laohekou
Frapp's Chemical (NFTZ) Co.,Ltd

Contact:+86-576-86137892

Address:General Chamber of Commercial Building, 159 Wanchang Middle Road, Wenling, Zhejiang, China
Beijing Mashi Fine Chemical Co.,Ltd.

Contact:+86-10-61271592

Address:Room 506, Section B, Kaichi Mansion, Industrial Development
sichuan tiancai fine co LTD.

website:http://www.tcfinechem.com/

Contact:18681346930

Address:baifu town,whou district
Zhejiang Chemicals Import & Export Corporation (ZHECHEM)

Contact:+86-571-87046953

Address:No. 37, Qingchun Road

Relevant to this article

Crystallographic study of a novel subnanomolar inhibitor provides insight on the binding interactions of alkenyldiarylmethanes with human immunodeficiency virus-1 reverse transcriptase

Doi:10.1021/jm901167t
(2009)
Transition metal-free, chemoselective arylation of thioamides yielding aryl thioimidates or N-aryl thioamides

Doi:10.1039/c8cc04795b
(2018)
Dehydration-type Ti-Claisen Condensation (Carbonhomologation) of α-Heteroatom-substituted Acetates with Alkyl Formates: Utilization as (Z)-Stereodefined Cross-coupling Partners and Application to Concise Synthesis of Strobilurin A

Doi:10.1002/adsc.201700879
(2017)
Effective and reversible DNA condensation induced by bifunctional molecules containing macrocyclic polyamines and naphthyl moieties

Doi:10.1016/j.bmc.2011.11.069
(2012)
D⁺-π-A^- charge-transfer molecules based on tricyanoquinodimethane and diphosphine metal complexes

Doi:10.1021/ic8008333
(2008)
Benzofused N-substituted cyclic enediynes: Activation and DNA-cleavage potential

Doi:10.1016/j.bmc.2008.02.044
(2008)

Article Doi