Journal of Medicinal Chemistry p. 5080 - 5095 (2019)
Update date:2022-08-15
Topics:
Fujimoto, Kazuki
Matsuoka, Eriko
Asada, Naoya
Tadano, Genta
Yamamoto, Takahiko
Nakahara, Kenji
Fuchino, Kouki
Ito, Hisanori
Kanegawa, Naoki
Moechars, Diederik
Gijsen, Harrie J. M.
Kusakabe, Ken-Ichi
BACE1 inhibitors hold potential as agents in disease-modifying treatment for Alzheimer's disease. BACE2 cleaves the melanocyte protein PMEL in pigment cells of the skin and eye, generating melanin pigments. This role of BACE2 implies that nonselective and
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