SYNTHETIC STUDIES ON TELEOCIDIN I. REGIOSELECTIVE INTRODUCTION OF 4-AMINO AND 7-ACYL GROUPS ON INDOLE DERIVATIVE

DOI: 10.1016/S0040-4039(00)94266-7

Source and publish data:

Tetrahedron Letters p. 4327 - 4330 (1986)

Update date:2022-07-29

Topics:

Authors:

Nakatsuka, Shin-ichi

Masuda, Toshiya

Asano, Osamu

Teramae, Tomohiro

Goto, Toshio

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Article abstract of DOI:10.1016/S0040-4039(00)94266-7

Nitration of indole-3-carboxylic esters, 3 and 9, afforded 4-nitro derivatives, 4 and 10. 10 was regioselectively derived to 15, which contains substituents at 4- and 7-positions of indole nucleus similary to teleocidins.

Full text of DOI:10.1016/S0040-4039(00)94266-7

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