SYNTHETIC STUDIES ON TELEOCIDIN I. REGIOSELECTIVE INTRODUCTION OF 4-AMINO AND 7-ACYL GROUPS ON INDOLE DERIVATIVE

DOI: 10.1016/S0040-4039(00)94266-7

Source and publish data:

Tetrahedron Letters p. 4327 - 4330 (1986)

Update date:2022-07-29

Topics:

Authors:

Nakatsuka, Shin-ichi

Masuda, Toshiya

Asano, Osamu

Teramae, Tomohiro

Goto, Toshio

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)94266-7

Nitration of indole-3-carboxylic esters, 3 and 9, afforded 4-nitro derivatives, 4 and 10. 10 was regioselectively derived to 15, which contains substituents at 4- and 7-positions of indole nucleus similary to teleocidins.

Full text of DOI:10.1016/S0040-4039(00)94266-7

Products guided by the article

Product name:1H-Indole-3-carboxylic acid, 4-nitro-, methyl ester

Cas No:109175-08-8

R&D Labs maybe for 109175-08-8

jiangsu senxuan pharmaceutical and chemical co.,ltd

Contact:86-523-87982810

Address:hongqiao industrial zone,taixing,jiangsu china
Beijing Zhongshuo Pharmaceutical T & D Co.,Ltd

Contact:0086-10-64430626

Address:ea No 16, HEPINGLI,DONGCHENG DISTRICT,BEIJING,P.R.CHINA.
Zhejiang Rongkai Chemical Technology Co.,Ltd.

Contact:+86-578-8185786

Address:Shangjiang Industrial Zone,Suichang
Shaanxi Lighte Optoelectronics Material Co., Ltd.

Contact:+86-29-88320728-622/619/620

Address:No.55 INDUSTRY ROAD 2,XI'AN NATIONAL CIVIL AEROSPACE INDUSTRIAL PARK.XI'AN China 710065.
Chongqing Changfeng Chemical Co., Ltd.

website:http://www.changfengchem.com

Contact:+86-23-67896333

Address:30th Floor, Longhu Ziduxingzuo Building A, 1st Branch,YuSong Rd., Yubei District, Chongqing, China

Relevant to this article

Doi:10.1021/ja01550a036
(1958)
Synthesis of novel enantiopure biphenyl P,N-ligands and application in palladium-catalyzed asymmetric addition of arylboronic acids to N-benzylisatin

Doi:10.1021/jo802036m
(2009)
Hypervalent iodine in synthesis XV: A convenient new method for the preparation of unsymmetrical diaryl selenides

Doi:10.1080/00397919408011497
(1994)
Novel 3,4-Diarylpyrrolidine-Based Chiral Ligands for the Asymmetric Reaction of Arylmagnesium Bromides with Aldehydes

Doi:10.1246/cl.1987.65
(1987)
A Selective Prostaglandin E₂ Receptor Subtype 2 (EP2) Antagonist Increases the Macrophage-Mediated Clearance of Amyloid-Beta Plaques

Doi:10.1021/acs.jmedchem.5b00567
(2015)
Bronsted acid catalyzed enantioselective three-component reaction involving the α addition of isocyanides to imines

Doi:10.1002/anie.200902385
(2009)

Article Doi