Organic Process Research and Development p. 557 - 561 (2018)
Update date:2022-08-03
Topics: Characterization Reaction Conditions Reaction Mechanism Work-up and purification Iterative Optimization Catalyst and Ligand Selection
Wu, Quanbing
Xiong, Xin
Cao, Yudong
He, Lijuan
Fei, Zhongbo
Two convergent syntheses for compound 1 are described that apply Buchwald-Hartwig coupling as the key step. This development work provides a direct comparison of the coupling results from different coupling partners and illustrates that more efficiency ca
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Doi:10.1055/s-1987-27915
(1987)Doi:10.1016/S0957-4166(98)00137-2
(1998)Doi:10.1016/S0040-4039(00)93604-9
(1991)Doi:10.1021/ja00212a051
(1988)Doi:10.1016/S0277-5387(00)81099-2
(1987)Doi:10.1002/ejoc.200800790
(2008)