Imidazo[2,1-b]thiazoles: Multitargeted inhibitors of both the insulin-like growth factor receptor and members of the epidermal growth factor family of receptor tyrosine kinases

DOI: 10.1016/j.bmcl.2010.03.015

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 2452 - 2455 (2010)

Update date:2022-08-02

Topics:

Authors:

Fidanze, Steve D.

Erickson, Scott A.

Wang, Gary T.

Mantei, Robert

Clark, Richard F.

Sorensen, Bryan K.

Bamaung, Nwe Y.

Kovar, Peter

Johnson, Eric F.

Swinger, Kerren K.

Stewart, Kent D.

Zhang, Qian

Tucker, Lora A.

Pappano, William N.

Wilsbacher, Julie L.

Wang, Jieyi

Sheppard, George S.

Bell, Randy L.

Davidsen, Steven K.

Hubbard, Robert D.

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Article abstract of DOI:10.1016/j.bmcl.2010.03.015

The design and enzyme activities of a novel class of imidazo[2,1-b]thiazoles is presented.

Full text of DOI:10.1016/j.bmcl.2010.03.015

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