Trifluoromethyl-substituted pyridyl- and pyrazolylboronic acids and esters: Synthesis and Suzuki-Miyaura cross-coupling reactions

DOI: 10.1039/b901024f

Source and publish data:

Organic and Biomolecular Chemistry p. 2155 - 2161 (2009)

Update date:2022-08-03

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Authors:

Clapham, Kate M.

Batsanov, Andrei S.

Bryce, Martin R.

Tarbit, Brian

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Article abstract of DOI:10.1039/b901024f

The synthesis of trifluoromethyl-substituted pyridylboronic acids and pyrazolylboronic esters is described via lithiation-boronation protocols (Schemes 1, 3 and 4). A study of their palladium-catalysed cross-couplings with heteroaryl halides is presented.

Full text of DOI:10.1039/b901024f

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