A NOVEL SHORT AND EFFICIENT ASYMMETRIC SYNTHESIS OF STATINE ANALOGUES

DOI: 10.1016/S0040-4039(00)86044-X

Source and publish data:

Tetrahedron Letters p. 2307 - 2310 (1988)

Update date:2022-08-02

Topics:

Authors:

Devant, Ralf M.

Radunz, Hans-E.

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Article abstract of DOI:10.1016/S0040-4039(00)86044-X

The statine analogues 1a-c have been obtained in high optical purity via addition of chiral acetate enolate 4 to the α-aminoaldehydes 5a-c, followed by transesterification.

Full text of DOI:10.1016/S0040-4039(00)86044-X

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