IODOCYCLISATIONS OF ALLYL-AMIDINES AND -UREAS

DOI: 10.1016/0040-4039(88)85071-8

Source and publish data:

Tetrahedron Letters p. 3001 - 3002 (1988)

Update date:2022-08-02

Topics: Nucleophilic substitution Mechanistic Studies Hypervalent Iodine Reagents Chemical Reaction Experimental conditions Synthetic Methodology Iodocyclization

Authors:

Hunt, Peter A.

May, Christopher

Moody, Christopher J.

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Article abstract of DOI:10.1016/0040-4039(88)85071-8

Iodocyclisation of allyl-amidines (1) and -ureas (4) gives imidazolines (2) and imidazolinones (5) respectively; in contrast, bromocyclisation of the amidine (1a) results in formation of the six-membered ring (3).

Full text of DOI:10.1016/0040-4039(88)85071-8

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