Synthesis of some conformationally restricted analogues of fentanyl

DOI: 10.1021/jm00214a035

Source and publish data:

Journal of Medicinal Chemistry p. 600 - 602 (1977)

Update date:2022-08-03

Topics:

Authors:

Berger Berger

Davidson

Langford

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Article abstract of DOI:10.1021/jm00214a035

The preparation of cis- and trans-2,3,4,4a,5,9b-hexahydro-2-phenethyl-5-propionyl-1H-pyrido[4,3-b]indole is described. These compounds, which are conformationally restricted analogues of the potent analgesic fentanyl, were devoid of analgesic or CNS activ

Full text of DOI:10.1021/jm00214a035

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