Tetrahedron Letters p. 3219 - 3222 (1988)
Update date:2022-07-31
Topics:
Lever, Susan Z.
Baidoo, Kwamena E.
Kramer, Alfred V.
Burns, H. Donald
A novel bifunctional chelate, 1, was designed and synthesized for the facile and efficient incorporation of technetium-99m into biomolecules under mild conditions.The agent features a thiolactone moiety which upon direct protein coupling via amine residue
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