A Facile Synthesis of 2-Substituted Azetidines

DOI: 10.1246/bcsj.61.3029

Source and publish data:

Bulletin of the Chemical Society of Japan p. 3029 - 3032 (1988)

Update date:2022-08-04

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Authors:

Shono, Tatsuya

Matsumura, Yoshihiro

Uchida, Kenshi

Nakatani, Fumihiko

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Article abstract of DOI:10.1246/bcsj.61.3029

A new method for the synthesis of 2-substituted azetidines has been exploited.The method consists of (1) anodic acetoxylation of 1-(p-tolylsulfonyl)azetidine at the 2-position and (2) subsequent nucleophilic substitution of the acetoxyl group with nucleophiles such as trimethylsilyl cyanide, allyltrimethylsilane, 2-acetoxyfuran, and trimethyl phosphite.

Full text of DOI:10.1246/bcsj.61.3029

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Product name:2-acetoxy-1-(p-tolylsulfonyl)azetidine

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