A Facile Synthesis of 2-Substituted Azetidines

DOI: 10.1246/bcsj.61.3029

Source and publish data:

Bulletin of the Chemical Society of Japan p. 3029 - 3032 (1988)

Update date:2022-08-04

Topics:

Authors:

Shono, Tatsuya

Matsumura, Yoshihiro

Uchida, Kenshi

Nakatani, Fumihiko

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1246/bcsj.61.3029

A new method for the synthesis of 2-substituted azetidines has been exploited.The method consists of (1) anodic acetoxylation of 1-(p-tolylsulfonyl)azetidine at the 2-position and (2) subsequent nucleophilic substitution of the acetoxyl group with nucleophiles such as trimethylsilyl cyanide, allyltrimethylsilane, 2-acetoxyfuran, and trimethyl phosphite.

Full text of DOI:10.1246/bcsj.61.3029

Products guided by the article

Product name:2-acetoxy-1-(p-tolylsulfonyl)azetidine

Cas No:119345-92-5

R&D Labs maybe for 119345-92-5

NEW FORTUNE INDUSTRIAL CO.,LTD.

website:http://newfortune.lookchem.com/

Contact:+86-25-8645-9456

Address:C4-105 GREEN ISLAND FLOWER TOWN
Zhejiang kehong chemical co., ltd

Contact:0086-575-85522000

Address:xiner center RD binhai industrial zone shaoxing zhejiang province P.R.China,312073
Goldwills Pharmaceuticals Co., Ltd.

Contact:0916-2237889 13991621155

Address:North Suburb of Hanzhong city, Shaanxi Province
Cangzhou Senary Chemical Science-tech Co., Ltd

Contact:+86-317-3563899, 3563699

Address:168 Jinde Road, Cangzhou, Hebei, China
TIC Gums, Inc.

Contact:410-273-7300; 800-221-3953

Address:4609 Richlynn Dr., PO Box 369, Belcamp, MD, 21017-0369, USA

Relevant to this article

A convenient synthesis of substituted 3-bromotetrahydrofurans from homoallylic alcohols

Doi:10.1016/j.tetlet.2004.10.013
(2004)
Palladium Assisted Transfer Hydrogenation of Cyclic α,β-Unsaturated Ketones by Ammonium Formate

Doi:10.1016/0040-4039(94)88193-6
(1994)
Synthesis of 4-Substituted Prolines as Conformationally Constrained Amino Acid Analogues

Doi:10.1021/jo00269a022
(1989)
Organocatalytic enantioselective cascade michael-michael-wittig reactions of phosphorus ylides: One-pot synthesis of the all-cis trisubstituted cyclohexenecarboxylates via the [1+2 + 3] annulation

Doi:10.1021/ol9021832
(2009)
γ-Fe₂O₃@SiO₂@4-(sulfoamino)butanoic acid as a novel superparamagnetic nanocatalyst promoted green synthesis of 5-(aryl)-5H-spiro[diindeno[1,2-b:2′,1′-e]pyridine-11,3′-indoline]-2′,10,12-trione derivatives

Doi:10.1007/s11164-018-3571-1
(2018)
Design, Synthesis, Antifungal Activities and SARs of (R)-2-Aryl-4,5-dihydrothiazole-4-carboxylic Acid Derivatives

Doi:10.1002/cjoc.201500619
(2015)

Article Doi