One-pot N-alkylation/Heck approach to substituted indoles

DOI: 10.1016/j.tetlet.2009.09.144

Source and publish data:

Tetrahedron Letters p. 6968 - 6972 (2009)

Update date:2022-08-04

Topics:

Authors:

Weinrich, Melissa L.

Beck, Hilary P.

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Article abstract of DOI:10.1016/j.tetlet.2009.09.144

Here, we report the palladium-catalyzed one-pot N-alkylation/Heck cyclization of anilines to substituted indoles employing Pd(OAc)₂/XPhos. The scope and limitations of this methodology will be described.

Full text of DOI:10.1016/j.tetlet.2009.09.144

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