Quinoxalin-2-carboxamides: Synthesis and pharmacological evaluation as serotonin type-3 (5-HT3) receptor antagonists

DOI: 10.3109/14756366.2010.543419

Source and publish data:

Journal of Enzyme Inhibition and Medicinal Chemistry p. 610 - 615 (2011)

Update date:2022-08-04

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Authors:

Mahesh, Radhakrishnan

Devadoss, Thangaraj

Pandey, Dilip Kumar

Yadav, Shushil Kumar

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Article abstract of DOI:10.3109/14756366.2010.543419

A series of quinoxalin-2-carboxamides were designed as per the pharmacophoric requirements of 5-HT₃ receptor antagonists and synthesized by condensing the carboxylic group of quinoxalin-2-carboxylic acid with various amines in the presence of 1

Full text of DOI:10.3109/14756366.2010.543419

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