MedChemComm p. 1054 - 1064 (2015)
Update date:2022-08-02
Topics:
Williams, Jodi T.
Gatfield, John
Roch, Catherine
Treiber, Alexander
Jenck, Francois
Bolli, Martin H.
Brotschi, Christine
Sifferlen, Thierry
Heidmann, Bibia
Boss, Christoph
Starting from a thienopiperidine lead compound with high intrinsic clearance in rat and human liver microsomes and low aqueous solubility, a novel series of 1-acyl-2-benzylpyrrolidines were discovered as potent and competitive dual orexin receptor antagon
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