Journal of Medicinal Chemistry p. 695 - 710 (2018)
Update date:2022-08-15
Topics:
Mazur, Marzena
Olczak, Jacek
Olejniczak, Sylwia
Koralewski, Robert
Czestkowski, Wojciech
Jedrzejczak, Anna
Golab, Jakub
Dzwonek, Karolina
Dymek, Barbara
Sklepkiewicz, Piotr L.
Zagozdzon, Agnieszka
Noonan, Tom
Mahboubi, Keyvan
Conway, Bruce
Sheeler, Ryan
Beckett, Paul
Hungerford, William M.
Podjarny, Alberto
Mitschler, Andre
Cousido-Siah, Alexandra
Fadel, Firas
Golebiowski, Adam
This article highlights our work toward the identification of a potent, selective, and efficacious acidic mammalian chitinase (AMCase) inhibitor. Rational design, guided by X-ray analysis of several inhibitors bound to human chitotriosidase (hCHIT1), led
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