Journal of Medicinal Chemistry p. 1330 - 1347 (2019)
Update date:2022-08-15
Topics:
Saccoliti, Francesco
Madia, Valentina Noemi
Tudino, Valeria
De Leo, Alessandro
Pescatori, Luca
Messore, Antonella
De Vita, Daniela
Scipione, Luigi
Brun, Reto
Kaiser, Marcel
M?ser, Pascal
Calvet, Claudia M.
Jennings, Gareth K.
Podust, Larissa M.
Pepe, Giacomo
Cirilli, Roberto
Faggi, Cristina
Di Marco, Annalise
Battista, Maria Rosaria
Summa, Vincenzo
Costi, Roberta
Di Santo, Roberto
We have designed and synthesized a series of new imidazole-based compounds structurally related to an antiprotozoal agent with nanomolar activity which we identified recently. The new analogues possess micromolar activities against Trypanosoma brucei rhod
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Doi:10.3184/030823410X12746990145128
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