
Journal of Medicinal Chemistry p. 1756 - 1764 (1990)
Update date:2022-08-05
Topics:
Brewster, William K.
Nichols, David E.
Riggs, Robert M.
Mottola, David M.
Lovenberg, Timothy W.
et al.
trans-10,11-Dihydroxy-5,6,6a,7,8,12b-hexahydrobenzophenanthridine (4a, dihydrexidine) has been found to be a highly potent and selective agonist of the dopamine D1 receptor in rat brain.Dihydrexidine had an EC50 of approximately 7
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