Bioorganic and Medicinal Chemistry Letters p. 3258 - 3261 (2007)
Update date:2022-09-26
Topics:
Denonne, Frederic
Binet, Sophie
Burton, Maggi
Collart, Philippe
Dipesa, Alan
Ganguly, Tanmoy
Giannaras, Alexander
Kumar, Seema
Lewis, Timothy
Maounis, Florence
Nicolas, Jean-Marie
Mansley, Tamsin
Pasau, Patrick
Preda, Dorin
Stebbins, Karin
Volosov, Alexander
Zou, Dong
The synthesis and in vitro binding of several new arginine-containing C3aR ligands are reported. DMPK properties and functional activities of selected compounds have been evaluated. One compound is shown to be active in an in vivo model of airway inflamma
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