Journal of Medicinal Chemistry p. 2259 - 2264 (1990)
Update date:2022-08-04
Topics:
Shyam
Penketh
Divo
Loomis
Patton
Sartorelli
Several 1,2,2-tris(sulfonyl)hydrazines, conceived as prodrugs of 1,2-bis(sulfonyl)hydrazines, were synthesized and evaluated for antineoplastic and trypanocidal activities in mice. 1-Methyl-1,2,2-tris(methylsulfonyl)hydrazine emerged as an extremely effic
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Doi:10.1021/ja00397a053
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