European Journal of Medicinal Chemistry p. 208 - 222 (2018)
Update date:2022-08-05
Topics:
Singh, L. Ravithej
Kumar, Ajeet
Upadhyay, Akanksha
Gupta, Sampa
Palanati, Gopala Reddy
Sikka, Kamakshi
Siddiqi, Mohammad Imran
Yadav, Prem N.
Sashidhara, Koneni V.
In this study, we presented rational designing and synthesis of coumarin-dihydroquinazolinone conjugates to evaluate their agonist activity at GPR109a receptor. Among the synthesized small molecule library, compound 10c displayed robust agonist action at
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