Boc-CCK-4 derivatives containing side-chain ureas as potent and selective CCK-A receptor agonists

DOI: 10.1021/jm00113a023

Source and publish data:

Journal of Medicinal Chemistry p. 2837 - 2842 (1991)

Update date:2022-07-29

Topics:

Authors:

Shiosaki

Lin Lin

Kopecka Kopecka

Tufano Tufano

Bianchi Bianchi

Miller Miller

Witte Witte

Nadzan Nadzan

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Article abstract of DOI:10.1021/jm00113a023

Novel Boc-CCK-4 derivatives were communicated recently as having high potency and selectivity for the CCK-A receptor (Shiosaki et al. J. Med. Chem. 1990, 33, 2950-2952). While Boc-CCK-4 binds selectively to the CCK-B receptor, replacement of the methionin

Full text of DOI:10.1021/jm00113a023

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