Synthesis and antiviral and cytostatic properties of 3'-deoxy-3'-fluoro- and 2'-azido-3'-fluoro-2',3'-dideoxy-D-ribofuranosides of natural heterocyclic bases

DOI: 10.1021/jm00111a040

Source and publish data:

Journal of Medicinal Chemistry p. 2195 - 2202 (1991)

Update date:2022-08-02

Topics:

Authors:

Mikhailopulo

Poopeiko

Pricota Pricota

Sivets Sivets

Kvasyuk Kvasyuk

Balzarini

De Clercq

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Article abstract of DOI:10.1021/jm00111a040

A series of 3'-deoxy-3'-fluoro- and 2'-azido-2',3'-dideoxy-3'-fluoro-D-ribofuranosides of natural heterocyclic bases have been synthesized with the use of universal carbohydrate precursors, viz., 1-O-acetyl-2,5-di-O-benzoyl-3-deoxy-3-fluoro-D-ribofuranose

Full text of DOI:10.1021/jm00111a040

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