Bioorganic and Medicinal Chemistry Letters p. 6782 - 6787 (2011)
Update date:2022-08-03
Topics:
Szabo, Monika
Agostino, Mark
Malone, Daniel T.
Yuriev, Elizabeth
Capuano, Ben
We have synthesised an extensive series of URB602 analogues as inhibitors of monoacylglycerol lipase (MAGL), which is the major enzyme responsible for metabolising the endocannabinoid 2-arachidonylglycerol. The recently identified crystal structure of MAG
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