Bioorganic and Medicinal Chemistry Letters p. 6782 - 6787 (2011)
Update date:2022-08-03
Topics:
Szabo, Monika
Agostino, Mark
Malone, Daniel T.
Yuriev, Elizabeth
Capuano, Ben
We have synthesised an extensive series of URB602 analogues as inhibitors of monoacylglycerol lipase (MAGL), which is the major enzyme responsible for metabolising the endocannabinoid 2-arachidonylglycerol. The recently identified crystal structure of MAG
View MoreGoldwills Pharmaceuticals Co., Ltd.
Contact:0916-2237889 13991621155
Address:North Suburb of Hanzhong city, Shaanxi Province
Chengdu D-Innovation Pharmaceutical Co., Ltd
Contact:86-28-85105536
Address:1001, B6, No.88 Keyuan South Road, Chengdu Hi-Tech Zone
Qingdao Pana-Life Biochem Co.,Ltd.
Contact:86-532-87683902
Address:No.967 Dalao Road, Licang Zone, Qingdao City,Shandong, China 266021
Suzhou Time-chem Technologies Co., Ltd.
Contact:0512-63983931/68086856
Address:No. 1326 of Binhe Road, New District, Suzhou, Jiangsu, P. R. China
WUHU HUAHAI BIOLOGY ENGINEERING CO LTD
Contact:+86-553-3836920
Address:7/F NO.82 LAODONG ROAD WUHU CHINA
Doi:10.1021/acs.orglett.6b01134
(2016)Doi:10.1007/s11164-017-2932-5
(2017)Doi:10.1016/S0040-4020(01)89562-4
(1994)Doi:10.1016/j.molstruc.2011.08.033
(2011)Doi:10.1080/15533174.2011.591353
(2011)Doi:10.1016/S0040-4039(00)74785-X
(1992)